Copper-catalyzed conversion of aryl and heteroaryl bromides into the corresponding chlorides.

نویسندگان

  • Xiujuan Feng
  • Yiping Qu
  • Yanlei Han
  • Xiaoqiang Yu
  • Ming Bao
  • Yoshinori Yamamoto
چکیده

An efficient method for the synthesis of aryl and heteroaryl chlorides is described. The reactions of aryl and heteroaryl bromides with tetramethylammonium chloride proceeded smoothly in the presence of a copper catalyst under mild reaction conditions to produce the corresponding chlorides in satisfactory to excellent yields.

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عنوان ژورنال:
  • Chemical communications

دوره 48 76  شماره 

صفحات  -

تاریخ انتشار 2012